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赵世振
2018-04-08 15:09  
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(信息截止2018年3月31日)

1、个人简介:

姓名:赵世振

学历:博士

政治面貌:中共党员

教育背景:

2007.9-2011.6 泰山医学院 专业:中药学 学士

2011.9-2014.6 沈阳药科大学 专业:药物化学 硕士

2014.9-2017.6 沈阳药科大学 专业:药物化学 博士

2、主要研究方向:

基于靶点的药物设计、合成及生物活性评价工作

3、已发表论文:

1)Shizhen Zhao, Liyu Zhao, Xiangqian Zhang, Chunchi Liu, Chenzhou Hao, Honglei Xie, Bin Sun, Dongmei Zhao*, Maosheng Cheng. Design, synthesis, and structure-activity relationship studies of benzothiazole derivatives as antifungal agents.[J].European Journal of Medicinal Chemistry, 2016, 123:514-522.

2)Shizhen Zhao, Xiangqian,PengWei, Xin Su, Liyu Zhao, Mengya Wu, Chenzhou Hao, Chunchi Liu, Dongmei Zhao*, Maosheng Cheng. Design, synthesis and evaluation of aromatic heterocyclic derivatives as potent antifungal agents[J].European Journal of Medicinal Chemistry, 2017, 137:96-107.

3)Dongmei Zhao*,Shizhen Zhao, Liyu Zhao, Xiangqian Zhang, Peng Wei, Chunchi Liu, Chenzhou Hao, Bin Sun, Xin Su*, Maosheng Cheng. Discovery of biphenyl imidazole derivatives as potent antifungal agents: Design, synthesis, and structure-activity relationship studies[J].Bioorganic & Medicinal Chemistry,2016, 25, 750-758.

4)Dongmei Zhao*, Honglei Xie, Changlin Bai, Chunchi Liu, Chenzhou Hao,Shizhen Zhao, Hongli Yuan, Changqun Luo, Jian Wang, Bin Lin, Jiang Zheng, Maosheng Cheng.Design, synthesis and biological evaluation of N,N-3-phenyl-3-benzylaminopropanamide derivatives as novel cholesteryl ester transfer protein inhibitor.[J].Bioorganic & Medicinal Chemistry, 2016, 24(8):1589-1597.

5)Chunchi Liu, Changqun Luo, Lijuan Hao, Qiong Wu, Honglei Xie,Shizhen Zhao, Chenzhou Hao, Dongmei Zhao*, Maosheng Cheng. Design, synthesis and biological evaluation of novel cholesteryl ester transfer protein inhibitors bearing a cycloalkene scaffold.[J].European Journal of Medicinal Chemistry, 2016, 123:419-430.

6)赵世振,赵冬梅*.氟班色林(Flibanserin)[J].中国药物化学杂志, 2016(1):82-82.

7)赵世振,谢洪磊,白长林,王凯,赵冬梅*.西沙比利合成工艺改进[J].中国药物化学杂志, 2016(2):116-119.

4、获得专利:

1)赵冬梅,孙彬,赵世振,程卯生,李凤荣,赵立雨,郝晨洲,刘春池,任金红.酰胺咪唑类衍生物及其用途[P].CN105541828A.

2)赵冬梅,赵世振,程卯生,赵立雨,张向前,魏鹏,吴梦雅,王德鑫.新型三环异恶唑类衍生物的制备方法及其在医药上的应用[P].CN201710422321.4.

3)李炳龙,刘常丽,赵世振,齐永秀,夏成才,李福荣,李珂,郝立勇,管西栋.一种由1,4二卤(异二卤)丁烷和甲硫醇钠合成4甲硫丁基硫氰酸酯的方法[P].CN106866478A.

5、联系方式(邮箱等):

E-mail:zhaoshizhen1987@163.com

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